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| 序号 | 结构式 | 产品名称 | KEY USE | ORIGINATOR |
| 31 | Finerenone 非奈利酮 |
Anti-diabetic nephropathy | BMS | |
| 32 | Lumateperone Tosylate 卢美哌隆对甲苯磺酸盐 |
Anti-schizophrenia | Janssen | |
| 33 | Apalutamide 阿帕鲁胺 |
Anti-prostatic cancer | Bayer | |
| 34 | Darolutamide 达洛鲁胺 |
Anti-prostatic cancer | Gilead | |
| 35 | Velpatasvir 维帕他韦 |
Anti-HCV | Shionogi | |
| 36 | Baloxavir Marboxil 玛巴洛沙韦 |
Anti-influenza | BMS | |
| 37 | Mavacamten 玛伐凯泰 |
Anti-HCM | BMS | |
| 38 | Rimegepant 瑞美吉泮 |
Anti-migraine | AbbVie | |
| 39 | Atogepant 阿托吉泮 |
Anti-migraine | Allergan | |
| 40 | Ubrogepant 乌布吉泮 |
Anti-migraine | Eli Lilly | |
| 41 | Lasmiditan Hemisuccinate 半琥珀酸拉米地坦 |
Anti-migraine | CJ HealthCare | |
| 42 | Tegoprazan 替格拉生 |
Gastroesphageal Reflux | Roche | |
| 43 | Resmetirom 瑞司美替罗 |
Anti-NASH | Blueprint Medicines | |
| 44 | Avapritinib 阿伐替尼 |
Anti-GIST | GBT | |
| 45 | Voxelotor 沃塞洛托 |
Anti-SCD | Novartis | |
| 46 | Iptacopan 盐酸伊普可泮 |
Anti-PNH | Novartis | |
| 47 | Atrasentan 阿曲生坦 |
Anti-nephropathy | Astellas | |
| 48 | Fezolinetant 非唑奈坦 |
Anti-VMS | Astellas | |
| 49 | Elinzanetant 依林奈坦 |
Anti-VMS | Bayer |